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TAK-802 hydrochloride

CAS No. 263248-36-8

TAK-802 hydrochloride( TAK 802 | TAK802 )

Catalog No. M13805 CAS No. 263248-36-8

A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM; exhibits high selectivity for acetylcholinesterase inhibition over butyrylcholinesterase inhibition.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    TAK-802 hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM; exhibits high selectivity for acetylcholinesterase inhibition over butyrylcholinesterase inhibition.
  • Description
    A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM; exhibits high selectivity for acetylcholinesterase inhibition over butyrylcholinesterase inhibition; increases rhythmic bladder contractions in Guinea pigs and rats without affecting the basal intravesical pressure.Other Indication Phase 2 Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    TAK 802 | TAK802
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    AChE
  • Recptor
    AChE
  • Research Area
    Other Indications
  • Indication
    Other Disease

Chemical Information

  • CAS Number
    263248-36-8
  • Formula Weight
    456.986
  • Molecular Formula
    C26H30ClFN2O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    8-[3-[1-[(3-fluorophenyl)methyl]-4-piperidinyl]-1-oxopropyl]-1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one hydrochloride

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ishichi Y, et al. Bioorg Med Chem. 2005 Mar 15;13(6):1901-11. 2. Nagabukuro H, et al. Eur J Pharmacol. 2004 Feb 6;485(1-3):299-305. 3. Nagabukuro H, et al. Eur J Pharmacol. 2004 Jun 28;494(2-3):225-32.
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